N-phenyl-N'-[4-(5H-pyrrolo[3,2-d]pyrimidin-4-yloxy)phenyl]ureas as novel inhibitors of VEGFR and FGFR kinases.
作者:
主题词
结合部位(Binding Sites);细胞, 培养的(Cells, Cultured);计算机模拟(Computer Simulation);结晶学, X线(Crystallography, X-Ray);药物设计(Drug Design);人类(Humans);苯脲化合物(Phenylurea Compounds);蛋白激酶抑制剂(Protein Kinase Inhibitors);嘧啶类(Pyrimidines);吡咯类(Pyrroles);受体, TIE-2(Receptor, TIE-2);受体, 成纤维细胞生长因子(Receptors, Fibroblast Growth Factor);受体, 血小板源生长因子(Receptors, Platelet-Derived Growth Factor);受体, 血管内皮生长因子(Receptors, Vascular Endothelial Growth Factor);构效关系(Structure-Activity Relationship);尿素(Urea)
DOI
10.1016/j.bmc.2010.08.042
PMID
20833551
发布时间
2016-11-25
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