4-[N-(substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII.
第一作者:
Jurgis,Sūdžius
第一单位:
Department of Organic Chemistry, Faculty of Chemistry, Vilnius University, Naugarduko 24, LT-03225 Vilnius, Lithuania.
作者:
主题词
结合部位(Binding Sites);量热法(Calorimetry);碳酸酐酶Ⅰ(Carbonic Anhydrase I);碳酸酐酶Ⅱ(Carbonic Anhydrase II);碳酸酐酶抑制剂(Carbonic Anhydrase Inhibitors);碳酸酐酶类(Carbonic Anhydrases);结晶学, X线(Crystallography, X-Ray);人类(Humans);蛋白质结构, 三级(Protein Structure, Tertiary);嘧啶类(Pyrimidines);重组蛋白质类(Recombinant Proteins);构效关系(Structure-Activity Relationship);磺胺类(Sulfonamides)
DOI
10.1016/j.bmc.2010.09.011
PMID
20889345
发布时间
2023-12-13
- 浏览18
相似文献
- 中文期刊
- 外文期刊
- 学位论文
- 会议论文