Small molecule AKAP-protein kinase A (PKA) interaction disruptors that activate PKA interfere with compartmentalized cAMP signaling in cardiac myocytes.
作者:
主题词
A型激酶锚定蛋白质类(A Kinase Anchor Proteins);别构调节(Allosteric Regulation);动物(Animals);慢性病(Chronic Disease);环AMP(Cyclic AMP);环AMP依赖性蛋白激酶类(Cyclic AMP-Dependent Protein Kinases);酶激活(Enzyme Activation);心力衰竭(Heart Failure);男(雄)性(Male);心肌收缩(Myocardial Contraction);肌细胞, 心脏(Myocytes, Cardiac);蛋白激酶抑制剂(Protein Kinase Inhibitors);大鼠(Rats);大鼠, 近交WKY(Rats, Inbred WKY);第二信使系统(Second Messenger Systems)
DOI
10.1074/jbc.M110.160614
PMID
21177871
发布时间
2024-06-07
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