Structure-activity studies of a novel series of isoxazole-3-carboxamide derivatives as TRPV1 antagonists.
作者:
主题词
酰胺类(Amides);动物(Animals);抗高血压药(Antihypertensive Agents);环己醇类(Cyclohexanols);高温, 诱发(Hyperthermia, Induced);异恶唑类(Isoxazoles);大鼠(Rats);大鼠, Wistar(Rats, Wistar);构效关系(Structure-Activity Relationship);TRPV阳离子通道(TRPV Cation Channels)
DOI
10.1016/j.bmcl.2010.12.092
PMID
21236666
发布时间
2011-01-24
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