Biochemical mechanism of pathogenesis of human gonadotropin-releasing hormone receptor mutants Thr104Ile and Tyr108Cys associated with familial hypogonadotropic hypogonadism.
作者:
主题词
结合, 竞争性(Binding, Competitive);布舍瑞林(Buserelin);细胞, 培养的(Cells, Cultured);剂量效应关系, 药物(Dose-Response Relationship, Drug);人类(Humans);性腺功能减退症(Hypogonadism);半数抑制浓度(Inhibitory Concentration 50);肌醇磷酸类(Inositol Phosphates);分子动力学模拟(Molecular Dynamics Simulation);突变, 误义(Mutation, Missense);蛋白质结合(Protein Binding);蛋白质相互作用域和基序(Protein Interaction Domains and Motifs);受体, LHRH(Receptors, LHRH)
DOI
10.1016/j.mce.2011.01.016
PMID
21277937
发布时间
2021-10-20
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