PTEN loss confers BRAF inhibitor resistance to melanoma cells through the suppression of BIM expression.
第一作者:
Kim H T,Paraiso
第一单位:
Department of Molecular Oncology, The Moffitt Cancer Center & Research Institute, University of South Florida College of Medicine, Tampa, Florida, USA.
作者:
主题词
细胞凋亡(Apoptosis);凋亡调节蛋白质类(Apoptosis Regulatory Proteins);细胞系, 肿瘤(Cell Line, Tumor);抗药性, 肿瘤(Drug Resistance, Neoplasm);人类(Humans);吲哚类(Indoles);黑色素瘤(Melanoma);膜蛋白质类(Membrane Proteins);突变(Mutation);PTEN磷酸水解酶(PTEN Phosphohydrolase);磷酸肌醇3-激酶类(Phosphatidylinositol 3-Kinases);蛋白激酶抑制剂(Protein Kinase Inhibitors);原癌基因蛋白质类(Proto-Oncogene Proteins);原癌基因蛋白质B-raf(Proto-Oncogene Proteins B-raf);原癌基因蛋白质c-akt(Proto-Oncogene Proteins c-akt);RNA, 小分子干扰(RNA, Small Interfering);磺胺类(Sulfonamides);增量调节(Up-Regulation)
DOI
10.1158/0008-5472.CAN-10-2954
PMID
21317224
发布时间
2022-03-11
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Cancer research
2750-60页
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