A novel small molecule antagonist of choline kinase-α that simultaneously suppresses MAPK and PI3K/AKT signaling.
第一作者:
B F,Clem
第一单位:
Department of Medicine, University of Louisville, Louisville, KY 40202, USA.
作者:
主题词
乙酰胺类(Acetamides);肌动蛋白类(Actins);动物(Animals);细胞膜(Cell Membrane);细胞增殖(Cell Proliferation);胆碱激酶(Choline Kinase);计算生物学(Computational Biology);酶抑制剂(Enzyme Inhibitors);细胞外信号调节MAP激酶类(Extracellular Signal-Regulated MAP Kinases);女(雌)性(Female);人类(Humans);MAP激酶信号系统(MAP Kinase Signaling System);小鼠(Mice);丝裂原激活蛋白激酶类(Mitogen-Activated Protein Kinases);模型, 分子(Models, Molecular);磷酸肌醇3-激酶类(Phosphatidylinositol 3-Kinases);磷酰化(Phosphorylation);磷酰胆碱(Phosphorylcholine);蛋白质构象(Protein Conformation);原癌基因蛋白质c-akt(Proto-Oncogene Proteins c-akt);原癌基因蛋白质类p21(ras)(Proto-Oncogene Proteins p21(ras));三唑类(Triazoles);异种移植模型抗肿瘤试验(Xenograft Model Antitumor Assays)
DOI
10.1038/onc.2011.51
PMID
21423211
发布时间
2021-10-20
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Oncogene
3370-80页
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