Antitumor and antiangiogenic activities of BMS-690514, an inhibitor of human EGF and VEGF receptor kinase families.
第一作者:
Tai W,Wong
第一单位:
Oncology Discovery, Discovery Chemistry, and Discovery Medicine and Clinical Pharmacology, Bristol-Myers Squibb Research, Princeton, NJ 08543, USA. tai.wong@bms.com
作者:
医学主题词
血管生成抑制剂(Angiogenesis Inhibitors);动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);细胞系(Cell Line);细胞增殖(Cell Proliferation);内皮细胞(Endothelial Cells);女(雌)性(Female);人类(Humans);小鼠(Mice);小鼠, 近交BALB C(Mice, Inbred BALB C);小鼠, 裸(Mice, Nude);肿瘤(Neoplasms);新生血管化, 病理性(Neovascularization, Pathologic);哌啶类(Piperidines);吡咯类(Pyrroles);受体, 血管内皮生长因子(Receptors, Vascular Endothelial Growth Factor);局部血流(Regional Blood Flow);信号传导(Signal Transduction);三嗪类(Triazines);异种移植模型抗肿瘤试验(Xenograft Model Antitumor Assays)
DOI
10.1158/1078-0432.CCR-10-3417
PMID
21531814
发布时间
2022-03-09
- 浏览30
Clinical cancer research
4031-41页
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