The design, synthesis and structure-activity relationships of novel isoindoline-based histone deacetylase inhibitors.
作者:
主题词
抗肿瘤药(Antineoplastic Agents);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物设计(Drug Design);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);组蛋白脱乙酰基酶1(Histone Deacetylase 1);组蛋白脱乙酰基酶抑制剂(Histone Deacetylase Inhibitors);人类(Humans);羟肟酸类(Hydroxamic Acids);异吲哚类(Isoindoles);分子结构(Molecular Structure);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2011.06.015
PMID
21742496
发布时间
2011-07-29
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