The hydrophobic amino acids in putative helix 8 in carboxy-terminus of histamine H(3) receptor are involved in receptor-G-protein coupling.
作者:
主题词
氨基酸序列(Amino Acid Sequence);氨基酸类(Amino Acids);细胞膜(Cell Membrane);环AMP(Cyclic AMP);流式细胞术(Flow Cytometry);GTP结合蛋白质类(GTP-Binding Proteins);HEK293细胞(HEK293 Cells);组胺(Histamine);组胺激动药(Histamine Agonists);人类(Humans);亲水和疏水相互作用(Hydrophobic and Hydrophilic Interactions);分子序列数据(Molecular Sequence Data);诱变, 定点(Mutagenesis, Site-Directed);突变(Mutation);哌啶类(Piperidines);质粒(Plasmids);蛋白质结合(Protein Binding);蛋白质结构, 二级(Protein Structure, Secondary);受体, 组胺H3(Receptors, Histamine H3);信号传导(Signal Transduction);构效关系(Structure-Activity Relationship);转染(Transfection)
DOI
10.1016/j.cellsig.2011.06.021
PMID
21749919
发布时间
2016-11-25
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Cellular signalling
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