Synthesis and characterization of tritylthioethanamine derivatives with potent KSP inhibitory activity.
第一作者:
Delany,Rodriguez
第一单位:
Department of Biology, New Mexico State University, Las Cruces, NM 88003, USA.
作者:
医学主题词
动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);细胞, 培养的(Cells, Cultured);半胱胺(Cysteamine);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);胚胎, 非哺乳动物(Embryo, Nonmammalian);人类(Humans);模型, 分子(Models, Molecular);分子结构(Molecular Structure);海胆纲(Sea Urchins);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmc.2011.07.054
PMID
21855351
发布时间
2025-05-29
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