Pyrazolo[1,5-a]pyrimidines, triazolo[1,5-a]pyrimidines and their tricyclic derivatives as corticotropin-releasing factor 1 (CRF₁) receptor antagonists.
作者:
主题词
动物(Animals);人类(Humans);动力学(Kinetics);男(雄)性(Male);蛋白质结合(Protein Binding);嘧啶类(Pyrimidines);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);受体, 促肾上腺皮质素释放激素(Receptors, Corticotropin-Releasing Hormone);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmc.2011.08.055
PMID
21930387
发布时间
2018-12-01
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