Pharmacokinetics and pharmacodynamics of TMC207 and its N-desmethyl metabolite in a murine model of tuberculosis.
作者:
主题词
ATP合成酶复合物(ATP Synthetase Complexes);动物(Animals);抗结核药(Antitubercular Agents);曲线下面积(Area Under Curve);细菌蛋白质类(Bacterial Proteins);生物转化(Biotransformation);集落计数, 微生物(Colony Count, Microbial);疾病模型, 动物(Disease Models, Animal);投药途径(Drug Administration Routes);用药计划表(Drug Administration Schedule);药物剂量计算(Drug Dosage Calculations);女(雌)性(Female);半衰期(Half-Life);人类(Humans);肺(Lung);男(雄)性(Male);小鼠(Mice);微生物敏感性试验(Microbial Sensitivity Tests);结核分枝杆菌(Mycobacterium tuberculosis);喹啉类(Quinolines);结核, 肺(Tuberculosis, Pulmonary)
DOI
10.1128/AAC.00720-11
PMID
22155815
发布时间
2021-10-21
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