A novel µ-conopeptide, CnIIIC, exerts potent and preferential inhibition of NaV1.2/1.4 channels and blocks neuronal nicotinic acetylcholine receptors.
作者:
主题词
氨基酸序列(Amino Acid Sequence);动物(Animals);芋螺毒素类(Conotoxins);芋螺属(Conus Snail);狗鱼科(Esocidae);女(雌)性(Female);HEK293细胞(HEK293 Cells);人类(Humans);男(雄)性(Male);小鼠(Mice);分子序列数据(Molecular Sequence Data);肌收缩(Muscle Contraction);肌, 骨骼(Muscle, Skeletal);烟碱拮抗剂(Nicotinic Antagonists);嗅神经(Olfactory Nerve);卵母细胞(Oocytes);肽类(Peptides);蛋白质构象(Protein Conformation);受体, 烟碱(Receptors, Nicotinic);坐骨神经(Sciatic Nerve);钠通道阻滞剂(Sodium Channel Blockers);钠通道(Sodium Channels);光滑爪蟾(Xenopus laevis)
DOI
10.1111/j.1476-5381.2012.01837.x
PMID
22229737
发布时间
2021-10-21
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