Design, synthesis and molecular docking studies of some novel spiro[indoline-3, 4'-piperidine]-2-ones as potential c-Met inhibitors.
第一作者:
Lianbao,Ye
第一单位:
School of Pharmaceutical Sciences, Southern Medical University, Guangzhou 510515, China. yelb7909@163.com
作者:
主题词
结合部位(Binding Sites);印迹法, 蛋白质(Blotting, Western);细胞增殖(Cell Proliferation);药物设计(Drug Design);药物发现(Drug Discovery);荧光共振能量转移(Fluorescence Resonance Energy Transfer);人类(Humans);半数抑制浓度(Inhibitory Concentration 50);模型, 分子(Models, Molecular);分子结构(Molecular Structure);哌啶类(Piperidines);蛋白激酶抑制剂(Protein Kinase Inhibitors);原癌基因蛋白质c-met(Proto-Oncogene Proteins c-met);胃肿瘤(Stomach Neoplasms);构效关系(Structure-Activity Relationship);肿瘤细胞, 培养的(Tumor Cells, Cultured)
DOI
10.1016/j.ejmech.2012.02.016
PMID
22381355
发布时间
2012-11-15
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