An antagonist of human protease activated receptor-2 attenuates PAR2 signaling, macrophage activation, mast cell degranulation, and collagen-induced arthritis in rats.
第一作者:
Rink-Jan,Lohman
第一单位:
Institute for Molecular Bioscience, The University of Queensland, Brisbane, Queensland, Australia.
作者:
医学主题词
投药, 口服(Administration, Oral);动物(Animals);关节炎, 实验性(Arthritis, Experimental);生物利用度(Biological Availability);细胞脱颗粒(Cell Degranulation);二肽类(Dipeptides);女(雌)性(Female);人类(Humans);异恶唑类(Isoxazoles);巨噬细胞活化(Macrophage Activation);男(雄)性(Male);肥大细胞(Mast Cells);模型, 生物学(Models, Biological);寡肽类(Oligopeptides);大鼠(Rats);大鼠, Wistar(Rats, Wistar);受体, PAR-2(Receptor, PAR-2);信号传导(Signal Transduction)
DOI
10.1096/fj.11-201004
PMID
22467762
发布时间
2012-06-29
- 浏览3
FASEB journal
2877-87页
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