Pharmacological characterization of A-960656, a histamine H₃ receptor antagonist with efficacy in animal models of osteoarthritis and neuropathic pain.
第一作者:
Marlon,Cowart
第一单位:
Department of Neuroscience Research, Abbott Laboratories, Abbott Park, IL 60064, United States. marlon.d.cowart@abbott.com
作者:
医学主题词
动物(Animals);苯并噻唑类(Benzothiazoles);细胞膜通透性(Cell Membrane Permeability);疾病模型, 动物(Disease Models, Animal);狗(Dogs);快速延迟整流钾通道(Ether-A-Go-Go Potassium Channels);HEK293细胞(HEK293 Cells);心脏(Heart);组胺H3拮抗剂(Histamine H3 Antagonists);人类(Humans);男(雄)性(Male);神经痛(Neuralgia);骨关节炎(Osteoarthritis);骨关节炎, 膝(Osteoarthritis, Knee);哒嗪类(Pyridazines);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);受体, 组胺H3(Receptors, Histamine H3);底物特异性(Substrate Specificity)
DOI
10.1016/j.ejphar.2012.03.048
PMID
22504024
发布时间
2014-11-20
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