PDE5 inhibitors, sildenafil and vardenafil, reverse multidrug resistance by inhibiting the efflux function of multidrug resistance protein 7 (ATP-binding Cassette C10) transporter.
第一作者:
Jun-Jiang,Chen
第一单位:
Department of Pharmaceutical Sciences, College of Pharmacy and Allied Health Professions, St John's University, Jamaica, New York, USA.
作者:
医学主题词
抗肿瘤药(Antineoplastic Agents);抗药性, 多药(Drug Resistance, Multiple);荧光抗体技术(Fluorescent Antibody Technique);HEK293细胞(HEK293 Cells);人类(Humans);咪唑类(Imidazoles);免疫印迹法(Immunoblotting);多药耐药相关蛋白质类(Multidrug Resistance-Associated Proteins);磷酸二酯酶5抑制剂(Phosphodiesterase 5 Inhibitors);哌嗪类(Piperazines);嘌呤类(Purines);砜类(Sulfones);三嗪类(Triazines)
DOI
10.1111/j.1349-7006.2012.02328.x
PMID
22578167
发布时间
2021-10-21
- 浏览23
Cancer science
1531-7页
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