Removal of the tag from His-tagged ILYd4, a human CD59 inhibitor, significantly improves its physical properties and its activity.
作者:
主题词
氨基酸序列(Amino Acid Sequence);动物(Animals);抗体, 单克隆(Antibodies, Monoclonal);抗体, 单克隆, 鼠源性(Antibodies, Monoclonal, Murine-Derived);抗肿瘤药(Antineoplastic Agents);细菌素类(Bacteriocins);化学疗法, 辅助(Chemotherapy, Adjuvant);药物设计(Drug Design);抗药性, 肿瘤(Drug Resistance, Neoplasm);药物稳定性(Drug Stability);组氨酸(Histidine);人类(Humans);白血病, 淋巴细胞, 慢性, B细胞(Leukemia, Lymphocytic, Chronic, B-Cell);淋巴瘤, B细胞(Lymphoma, B-Cell);溶解度(Solubility)
DOI
10.2174/138161212802430486
PMID
22642361
发布时间
2021-10-21
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Current pharmaceutical design
4187-96页
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