A novel series of G-quadruplex ligands with selectivity for HIF-expressing osteosarcoma and renal cancer cell lines.
作者:
主题词
抗肿瘤药(Antineoplastic Agents);碱性螺旋-环-螺旋转录因子类(Basic Helix-Loop-Helix Transcription Factors);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);成纤维细胞(Fibroblasts);G四链体(G-Quadruplexes);人类(Humans);缺氧诱导因子1, α亚基(Hypoxia-Inducible Factor 1, alpha Subunit);肾肿瘤(Kidney Neoplasms);配体(Ligands);分子结构(Molecular Structure);骨肉瘤(Osteosarcoma);启动区, 遗传(Promoter Regions, Genetic);RNA, 信使(RNA, Messenger);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2012.07.009
PMID
22889802
发布时间
2024-02-10
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