Inhibition of α-class cytosolic human carbonic anhydrases I, II, IX and XII, and β-class fungal enzymes by carboxylic acids and their derivatives: new isoform-I selective nanomolar inhibitors.
第一作者:
Mario,Sechi
第一单位:
Dipartimento di Chimica e Farmacia, Università di Sassari, Via Muroni 23/A, 07100 Sassari, Italy. mario.sechi@uniss.it
作者:
主题词
白色念珠菌(Candida albicans);碳酸酐酶抑制剂(Carbonic Anhydrase Inhibitors);碳酸酐酶类(Carbonic Anhydrases);羧酸类(Carboxylic Acids);新型隐球菌(Cryptococcus neoformans);剂量效应关系, 药物(Dose-Response Relationship, Drug);人类(Humans);分子结构(Molecular Structure);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2012.07.094
PMID
22901388
发布时间
2012-08-31
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