Selective histone deacetylase 6 inhibitors bearing substituted urea linkers inhibit melanoma cell growth.
第一作者:
Joel A,Bergman
第一单位:
Drug Discovery Program, Department of Medicinal Chemistry and Pharmacognosy, University of Illinois at Chicago, Chicago, Illinois 60612, USA.
作者:
主题词
乙酰化作用(Acetylation);动物(Animals);抗肿瘤药(Antineoplastic Agents);印迹法, 蛋白质(Blotting, Western);组蛋白脱乙酰基酶抑制剂(Histone Deacetylase Inhibitors);组蛋白脱乙酰基酶类(Histone Deacetylases);组蛋白类(Histones);人类(Humans);羟肟酸类(Hydroxamic Acids);同工酶类(Isoenzymes);黑色素瘤, 实验性(Melanoma, Experimental);小鼠(Mice);分子结构(Molecular Structure);苯脲化合物(Phenylurea Compounds);构效关系(Structure-Activity Relationship);肿瘤细胞, 培养的(Tumor Cells, Cultured);尿素(Urea)
DOI
10.1021/jm301098e
PMID
23009203
发布时间
2021-10-21
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