The inhibitor of Ca(2+)-dependent K+ channels TRAM-34 blocks growth of hepatocellular carcinoma cells via downregulation of estrogen receptor alpha mRNA and nuclear factor-kappaB.
作者:
主题词
细胞凋亡(Apoptosis);印迹法, 蛋白质(Blotting, Western);癌, 肝细胞(Carcinoma, Hepatocellular);细胞增殖(Cell Proliferation);雌激素受体α(Estrogen Receptor alpha);人类(Humans);瞬时电导钙激活钾通道(Intermediate-Conductance Calcium-Activated Potassium Channels);肝肿瘤(Liver Neoplasms);吡唑类(Pyrazoles);RNA, 信使(RNA, Messenger);RNA, 小分子干扰(RNA, Small Interfering);逆转录聚合酶链反应(Reverse Transcriptase Polymerase Chain Reaction);转录因子RelA(Transcription Factor RelA);肿瘤细胞, 培养的(Tumor Cells, Cultured)
DOI
10.1007/s10637-012-9879-6
PMID
23054207
发布时间
2021-10-21
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