Cerebrovascular dilation via selective targeting of the cholane steroid-recognition site in the BK channel β1-subunit by a novel nonsteroidal agent.
第一作者:
Anna N,Bukiya
第一单位:
Departments of Pharmacology, University of Tennessee Health Science Center, Memphis, TN 38163, USA.
作者:
主题词
动物(Animals);脑动脉(Cerebral Arteries);胆烷类(Cholanes);女(雌)性(Female);大电导钙激活钾通道β亚基(Large-Conductance Calcium-Activated Potassium Channel beta Subunits);石胆酸(Lithocholic Acid);男(雄)性(Male);小鼠(Mice);小鼠, 近交C57BL(Mice, Inbred C57BL);单核细胞(Monocytes);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);甾类(Steroids);血管舒张(Vasodilation);光滑爪蟾(Xenopus laevis)
DOI
10.1124/mol.112.083519
PMID
23455312
发布时间
2025-02-13
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Molecular pharmacology
1030-44页
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