Bcl-2/Bcl-xL inhibition increases the efficacy of MEK inhibition alone and in combination with PI3 kinase inhibition in lung and pancreatic tumor models.
第一作者:
Nguyen,Tan
第一单位:
Genentech, Inc., South San Francisco, CA 94080, USA.
作者:
医学主题词
苯胺化合物(Aniline Compounds);细胞凋亡(Apoptosis);细胞系, 肿瘤(Cell Line, Tumor);酶抑制剂(Enzyme Inhibitors);基因, bcl-2(Genes, bcl-2);人类(Humans);吲唑类(Indazoles);肺肿瘤(Lung Neoplasms);MAP激酶激酶激酶类(MAP Kinase Kinase Kinases);分子靶向治疗(Molecular Targeted Therapy);胰腺肿瘤(Pancreatic Neoplasms);磷酸肌醇3-激酶类(Phosphatidylinositol 3-Kinases);信号传导(Signal Transduction);磺胺类(Sulfonamides);bcl-X蛋白质(bcl-X Protein)
DOI
10.1158/1535-7163.MCT-12-0949
PMID
23475955
发布时间
2022-03-30
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