Synthesis and biological evaluation of urea derivatives as highly potent and selective rho kinase inhibitors.
作者:
主题词
腺苷三磷酸(Adenosine Triphosphate);动物(Animals);细胞系(Cell Line);人类(Humans);半数抑制浓度(Inhibitory Concentration 50);蛋白质构象(Protein Conformation);蛋白激酶抑制剂(Protein Kinase Inhibitors);大鼠(Rats);构效关系(Structure-Activity Relationship);底物特异性(Substrate Specificity);尿素(Urea);rho相关激酶类(rho-Associated Kinases)
DOI
10.1021/jm400062r
PMID
23570561
发布时间
2013-11-21
- 浏览36

Journal of medicinal chemistry
3568-81页
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