Inhibition of tumor angiogenesis and growth by a small-molecule multi-FGF receptor blocker with allosteric properties.
作者:
主题词
别构调节(Allosteric Regulation);动物(Animals);抗体, 单克隆(Antibodies, Monoclonal);关节炎, 实验性(Arthritis, Experimental);骨质吸收(Bone Resorption);癌, Lewis肺(Carcinoma, Lewis Lung);成纤维细胞生长因子(Fibroblast Growth Factors);HEK293细胞(HEK293 Cells);人类(Humans);小鼠(Mice);新生血管化, 病理性(Neovascularization, Pathologic);胰腺肿瘤(Pancreatic Neoplasms);磷酰化(Phosphorylation);蛋白激酶抑制剂(Protein Kinase Inhibitors);受体蛋白质酪氨酸激酶类(Receptor Protein-Tyrosine Kinases);受体, 成纤维细胞生长因子(Receptors, Fibroblast Growth Factor);信号传导(Signal Transduction);小分子化合物库(Small Molecule Libraries);异种移植模型抗肿瘤试验(Xenograft Model Antitumor Assays)
DOI
10.1016/j.ccr.2013.02.019
PMID
23597562
发布时间
2013-04-19
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Cancer cell
477-88页
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