Discovery of a novel ERK inhibitor with activity in models of acquired resistance to BRAF and MEK inhibitors.
作者:
主题词
细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);抗药性, 肿瘤(Drug Resistance, Neoplasm);细胞外信号调节MAP激酶类(Extracellular Signal-Regulated MAP Kinases);人类(Humans);MAP激酶激酶激酶类(MAP Kinase Kinase Kinases);突变(Mutation);肿瘤(Neoplasms);蛋白激酶抑制剂(Protein Kinase Inhibitors);原癌基因蛋白质B-raf(Proto-Oncogene Proteins B-raf);信号传导(Signal Transduction)
DOI
10.1158/2159-8290.CD-13-0070
PMID
23614898
发布时间
2013-07-12
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Cancer discovery
742-50页
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