Monitoring tumor response to linifanib therapy with SPECT/CT using the integrin αvβ3-targeted radiotracer 99mTc-3P-RGD2.
作者:
主题词
血管生成抑制剂(Angiogenesis Inhibitors);动物(Animals);二聚作用(Dimerization);女(雌)性(Female);神经胶质瘤(Glioma);人类(Humans);吲唑类(Indazoles);整合素αVβ3(Integrin alphaVbeta3);男(雄)性(Male);小鼠(Mice);小鼠, 裸(Mice, Nude);寡肽类(Oligopeptides);有机锝化合物(Organotechnetium Compounds);肽类, 环(Peptides, Cyclic);苯脲化合物(Phenylurea Compounds);正电子发射断层显像术(Positron-Emission Tomography);前列腺肿瘤(Prostatic Neoplasms);蛋白酪氨酸激酶类(Protein-Tyrosine Kinases);放射性药物(Radiopharmaceuticals);锝(Technetium);体层摄影术, X线计算机(Tomography, X-Ray Computed);异种移植模型抗肿瘤试验(Xenograft Model Antitumor Assays)
DOI
10.1124/jpet.112.202622
PMID
23750021
发布时间
2022-06-02
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