In vivo characterization of the highly selective monoacylglycerol lipase inhibitor KML29: antinociceptive activity without cannabimimetic side effects.
第一作者:
B M,Ignatowska-Jankowska
第一单位:
Department of Pharmacology and Toxicology, Virginia Commonwealth University, Richmond, VA, USA.
作者:
医学主题词
镇痛药(Analgesics);动物(Animals);消炎药, 非甾类(Anti-Inflammatory Agents, Non-Steroidal);苯并二恶茂类(Benzodioxoles);脑(Brain);大麻酚类(Cannabinoids);色谱法, 液相(Chromatography, Liquid);酶抑制剂(Enzyme Inhibitors);男(雄)性(Male);小鼠(Mice);小鼠, 近交C57BL(Mice, Inbred C57BL);分子模拟(Molecular Mimicry);单酰基甘油酯脂酶类(Monoacylglycerol Lipases);哌啶类(Piperidines);串联质谱法(Tandem Mass Spectrometry)
DOI
10.1111/bph.12298
PMID
23848221
发布时间
2024-04-20
- 浏览56
British journal of pharmacology
1392-407页
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