Discovery of N-(2,3,5-triazoyl)mycophenolic amide and mycophenolic epoxyketone as novel inhibitors of human IMPDH.
作者:
主题词
酰胺类(Amides);抗肿瘤药(Antineoplastic Agents);细胞分化(Cell Differentiation);细胞增殖(Cell Proliferation);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物发现(Drug Discovery);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);酶抑制剂(Enzyme Inhibitors);环氧化合物(Epoxy Compounds);人类(Humans);IMP脱氢酶(IMP Dehydrogenase);K562细胞(K562 Cells);酮类(Ketones);分子结构(Molecular Structure);构效关系(Structure-Activity Relationship);三唑类(Triazoles)
DOI
10.1016/j.bmcl.2013.07.016
PMID
23937979
发布时间
2013-08-23
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