Comparative analysis of ER stress response into HIV protease inhibitors: lopinavir but not darunavir induces potent ER stress response via ROS/JNK pathway.
第一作者:
Manabu,Taura
第一单位:
Division of Hematopoiesis, Center for AIDS Research, Kumamoto University, 2-2-1 Honjo, Kumamoto, 860-0811, Japan.
作者:
关键词
AIDSAPVAREATVAmprenavirAtazanavirCHOPCombination antiretroviral therapyDRVDarunavirER stressFDAFood and Drug AdministrationHIV protease inhibitorIDVIndinavirJNKLDHLPVLopinavirN-acetyl-L-cysteineNACNFVNelfinavirPBMCPIPRIPeripheral blood mononuclear cellsPropidium iodideProtease inhibitorROSRTVRitonavirSQVSaquinavirTPVTiprenavirantioxidant responsecARTlactate dehydrogenase
主题词
动物(Animals);细胞凋亡(Apoptosis);HEK293细胞(HEK293 Cells);HIV蛋白酶抑制药(HIV Protease Inhibitors);Hep G2细胞(Hep G2 Cells);人类(Humans);小肠(Intestine, Small);JNK丝裂原活化蛋白激酶类(JNK Mitogen-Activated Protein Kinases);肾(Kidney);肝(Liver);男(雄)性(Male);小鼠(Mice);小鼠, 近交BALB C(Mice, Inbred BALB C);活性氧(Reactive Oxygen Species);信号传导(Signal Transduction);磺胺类(Sulfonamides)
DOI
10.1016/j.freeradbiomed.2013.08.161
PMID
23973637
发布时间
2018-09-06
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Free radical biology & medicine
778-788页
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