Non-catalytic site HIV-1 integrase inhibitors disrupt core maturation and induce a reverse transcription block in target cells.
作者:
主题词
衔接蛋白质类, 信号转导(Adaptor Proteins, Signal Transducing);细胞系, 肿瘤(Cell Line, Tumor);DNA, 病毒(DNA, Viral);抗药性, 病毒(Drug Resistance, Viral);基因表达(Gene Expression);基因, 报告(Genes, Reporter);遗传载体(Genetic Vectors);HIV整合酶(HIV Integrase);HIV整合酶抑制剂(HIV Integrase Inhibitors);HIV逆转录酶(HIV Reverse Transcriptase);HIV-1(HIV-1);宿主与病原体相互作用(Host-Pathogen Interactions);人类(Humans);萤光素酶类(Luciferases);突变(Mutation);T淋巴细胞(T-Lymphocytes);转录因子(Transcription Factors);病毒粒子(Virion);病毒装配(Virus Assembly);病毒整合(Virus Integration);病毒复制(Virus Replication)
DOI
10.1371/journal.pone.0074163
PMID
24040198
发布时间
2021-10-21
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