Discovery of Small-Molecule Glucokinase Regulatory Protein Modulators That Restore Glucokinase Activity.
作者:
主题词
衔接蛋白质类, 信号转导(Adaptor Proteins, Signal Transducing);腺苷三磷酸(Adenosine Triphosphate);别构调节(Allosteric Regulation);动物(Animals);血糖(Blood Glucose);量热法(Calorimetry);糖尿病, 2型(Diabetes Mellitus, Type 2);药物发现(Drug Discovery);荧光(Fluorescence);荧光计(Fluorometry);果糖磷酸类(Fructosephosphates);葡糖激酶(Glucokinase);肝细胞(Hepatocytes);己糖磷酸盐类(Hexosephosphates);内环境稳定(Homeostasis);人类(Humans);低血糖症(Hypoglycemia);半数抑制浓度(Inhibitory Concentration 50);发光(Luminescence);蛋白质结合(Protein Binding);蛋白质构象(Protein Conformation);蛋白质相互作用图谱(Protein Interaction Mapping);大鼠(Rats);表面等离激元(Surface Plasmon Resonance)
DOI
10.1177/1087057114530468
PMID
24717911
发布时间
2016-12-30
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