Identification of neuropeptide S antagonists: structure-activity relationship studies, X-ray crystallography, and in vivo evaluation.
作者:
主题词
动物(Animals);CHO细胞(CHO Cells);仓鼠属(Cricetulus);结晶学, X线(Crystallography, X-Ray);人类(Humans);亲水和疏水相互作用(Hydrophobic and Hydrophilic Interactions);异构现象(Isomerism);男(雄)性(Male);小鼠, 近交C57BL(Mice, Inbred C57BL);分子结构(Molecular Structure);运动活动(Motor Activity);神经肽类(Neuropeptides);神经递质药(Neurotransmitter Agents);恶唑烷酮类(Oxazolidinones);吡嗪类(Pyrazines);受体, 神经肽(Receptors, Neuropeptide);溶解度(Solubility);构效关系(Structure-Activity Relationship);水(Water)
DOI
10.1021/cn500113c
PMID
24964000
发布时间
2024-05-07
- 浏览21

ACS chemical neuroscience
731-44页
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