Design, synthesis and pharmacological evaluation of novel polycyclic heteroarene ethers as PDE10A inhibitors: part II.
第一作者:
Sanjib,Das
第一单位:
Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
作者:
医学主题词
动物(Animals);狗(Dogs);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物设计(Drug Design);醚类(Ethers);直鼻猴亚目(Haplorhini);人类(Humans);男(雄)性(Male);小鼠(Mice);分子结构(Molecular Structure);磷酸二酯酶抑制剂(Phosphodiesterase Inhibitors);磷酸二酯水解酶类(Phosphoric Diester Hydrolases);吡嗪类(Pyrazines);吡啶类(Pyridines);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2014.06.028
PMID
24980052
发布时间
2014-07-11
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