A class of 4-sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects.
作者:
主题词
动物(Animals);二氧化碳(Carbon Dioxide);碳酸酐酶抑制剂(Carbonic Anhydrase Inhibitors);碳酸酐酶类(Carbonic Anhydrases);结晶学, X线(Crystallography, X-Ray);疾病模型, 动物(Disease Models, Animal);药物设计(Drug Design);醚类(Ethers);荧光染料(Fluorescent Dyes);青光眼(Glaucoma);人类(Humans);动力学(Kinetics);男(雄)性(Male);模型, 化学(Models, Chemical);分子结构(Molecular Structure);肿瘤(Neoplasms);兔(Rabbits);构效关系(Structure-Activity Relationship);水(Water)
DOI
10.1021/jm501497m
PMID
25358036
发布时间
2021-10-21
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