In vitro selective inhibition of human UDP-glucuronosyltransferase (UGT) 1A4 by finasteride, and prediction of in vivo drug-drug interactions.
第一作者:
Seung Jun,Lee
第一单位:
College of Pharmacy and Integrated Research Institute of Pharmaceutical Sciences, The Catholic University of Korea, 43 Jibong-ro, Wonmi-gu, Bucheon 420-743, Republic of Korea.
作者:
主题词
药物相互作用(Drug Interactions);酶抑制剂(Enzyme Inhibitors);非那特利(Finasteride);葡糖醛酸基转移酶(Glucuronosyltransferase);人类(Humans);同工酶类(Isoenzymes);动力学(Kinetics);微粒体, 肝(Microsomes, Liver);重组蛋白质类(Recombinant Proteins)
DOI
10.1016/j.toxlet.2014.11.018
PMID
25448279
发布时间
2019-03-28
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Toxicology letters
458-65页
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