Brain histamine H1 receptor occupancy measured by PET after oral administration of levocetirizine, a non-sedating antihistamine.
第一作者:
Kotaro,Hiraoka
第一单位:
Tohoku University, Cyclotron and Radioisotope Center, Division of Cyclotron Nuclear Medicine , 6-3, Aoba, Aramaki, Aoba-ku, Sendai, 980-8578 , Japan.
作者:
主题词
投药, 口服(Administration, Oral);脑(Brain);碳放射性同位素(Carbon Radioisotopes);西替利嗪(Cetirizine);交叉研究(Cross-Over Studies);双盲法(Double-Blind Method);多塞平(Doxepin);组胺H1拮抗剂, 非镇静(Histamine H1 Antagonists, Non-Sedating);人类(Humans);男(雄)性(Male);正电子发射断层显像术(Positron-Emission Tomography);放射配体测定(Radioligand Assay);受体, 组胺H1(Receptors, Histamine H1);睡眠(Sleep);特非那定(Terfenadine);青年人(Young Adult)
DOI
10.1517/14740338.2015.989831
PMID
25466429
发布时间
2015-11-19
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