IRS2 copy number gain, KRAS and BRAF mutation status as predictive biomarkers for response to the IGF-1R/IR inhibitor BMS-754807 in colorectal cancer cell lines.
第一作者:
Fei,Huang
第一单位:
Bristol-Myers Squibb Company, Princeton, New Jersey. fei.huang@bms.com han.chang@bms.com.
作者:
医学主题词
印迹法, 蛋白质(Blotting, Western);细胞系, 肿瘤(Cell Line, Tumor);结直肠肿瘤(Colorectal Neoplasms);DNA拷贝数变异(DNA Copy Number Variations);DNA突变分析(DNA Mutational Analysis);基因扩增(Gene Amplification);基因剂量(Gene Dosage);人类(Humans);胰岛素受体底物蛋白质类(Insulin Receptor Substrate Proteins);胰岛素样生长因子结合蛋白质6(Insulin-Like Growth Factor Binding Protein 6);配体(Ligands);模型, 生物学(Models, Biological);突变(Mutation);磷酰化(Phosphorylation);原癌基因蛋白质类(Proto-Oncogene Proteins);原癌基因蛋白质B-raf(Proto-Oncogene Proteins B-raf);原癌基因蛋白质类p21(ras)(Proto-Oncogene Proteins p21(ras));吡唑类(Pyrazoles);受体, IGF1型(Receptor, IGF Type 1);受体, 胰岛素(Receptor, Insulin);三嗪类(Triazines);ras蛋白质类(ras Proteins)
DOI
10.1158/1535-7163.MCT-14-0794-T
PMID
25527633
发布时间
2020-09-30
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