In vitro/in vivo investigations to examine the gender differences in the pharmacokinetics of novel oral Janus kinase (JAK) inhibitor ASP015K and sulfate metabolite M2 in rats.
第一作者:
Kazuo,Oda
第一单位:
Analysis & Pharmacokinetics Research Laboratories, Astellas Pharma Inc. , Yodogawa-ku, Osaka , Japan.
作者:
主题词
投药, 口服(Administration, Oral);动物(Animals);细胞色素P450酶系统(Cytochrome P-450 Enzyme System);女(雌)性(Female);Janus激酶类(Janus Kinases);男(雄)性(Male);蛋白激酶抑制剂(Protein Kinase Inhibitors);大鼠(Rats);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);性征(Sex Characteristics);磺基转移酶类(Sulfotransferases)
DOI
10.3109/00498254.2014.995747
PMID
25539455
发布时间
2015-07-03
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