Pharmacological evidence that histamine H3 receptors inhibit the vasodepressor responses by selective stimulation of the rat perivascular sensory CGRPergic outflow.
第一单位:
Departamento de Farmacobiología, Cinvestav-Coapa, Czda. Tenorios No. 235, Col. Granjas-Coapa, Deleg. Tlalpan, 14330 México D.F., Mexico. Electronic address: manriquegpe@yahoo.com.mx.
作者:
关键词
CGRPGallamine triethiodide (Pubchem CID: 6172)Hexamethonium chloride (Pubchem CID: 93550)Histamine receptorsImmepip dihydrobromide (Pubchem CID: 16078980)JNJ7777120 (Pubchem CID: 4908365)Ketotifen fumarate salt (Pubchem CID: 5282408)Methoxamine hydrochloride (Pubchem CID: 6081)Pithed ratRanitidine hydrochloride (Pubchem CID: 3033332)Sensory CGRPergic outflowThioperamide maleate salt (Pubchem CID: 16220001)α-CGRP (Pubchem CID: 56841902)
主题词
动物(Animals);血压(Blood Pressure);降钙素基因相关肽(Calcitonin Gene-Related Peptide);剂量效应关系, 药物(Dose-Response Relationship, Drug);电刺激(Electric Stimulation);心率(Heart Rate);组胺激动药(Histamine Agonists);组胺拮抗药(Histamine Antagonists);咪唑类(Imidazoles);男(雄)性(Male);哌啶类(Piperidines);大鼠(Rats);受体, 组胺H3(Receptors, Histamine H3);脊髓(Spinal Cord)
DOI
10.1016/j.ejphar.2015.02.017
PMID
25704614
发布时间
2018-12-02
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