Synthesis and Evaluation of 3-(furo[2,3-b]pyridin-3-yl)-4-(1H-indol-3-yl)-maleimides as Novel GSK-3β Inhibitors and Anti-Ischemic Agents.
第一作者:
Qing,Ye
第一单位:
State Key Laboratory Breeding Base of Green Chemistry-Synthesis Technology, Zhejiang University of Technology, Hangzhou, 310032, China.;State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
作者:
医学主题词
动物(Animals);脑缺血(Brain Ischemia);细胞, 培养的(Cells, Cultured);疾病模型, 动物(Disease Models, Animal);药物评价, 临床前(Drug Evaluation, Preclinical);酶抑制剂(Enzyme Inhibitors);谷氨酸(Glutamic Acid);糖原合成酶激酶3(Glycogen Synthase Kinase 3);半数抑制浓度(Inhibitory Concentration 50);马来酰亚胺类(Maleimides);神经元(Neurons);神经保护药(Neuroprotective Agents);大鼠(Rats);构效关系(Structure-Activity Relationship)
DOI
10.1111/cbdd.12546
PMID
25711384
发布时间
2016-11-25
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