Highly Selective Phosphatidylinositol 4-Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action.
第一作者:
Ivana,Mejdrová
第一单位:
‡Gilead Sciences, Inc., 333 Lakeside Drive, Foster City, California 94404, United States.
作者:
医学主题词
腺苷三磷酸(Adenosine Triphosphate);抗病毒药(Antiviral Agents);结合部位(Binding Sites);结晶学, X线(Crystallography, X-Ray);乙二胺类(Ethylenediamines);人类(Humans);咪唑类(Imidazoles);同工酶类(Isoenzymes);磷酸转移酶类(醇族体)(Phosphotransferases (Alcohol Group Acceptor));蛋白质构象(Protein Conformation);吡唑类(Pyrazoles);吡啶类(Pyridines);嘧啶类(Pyrimidines);RNA病毒(RNA Viruses);构效关系(Structure-Activity Relationship);三嗪类(Triazines)
DOI
10.1021/acs.jmedchem.5b00499
PMID
25897704
发布时间
2015-05-14
- 浏览36
Journal of medicinal chemistry
3767-93页
相似文献
- 中文期刊
- 外文期刊
- 学位论文
- 会议论文


换一批



