Structure-based drug design studies of the interactions of ent-kaurane diterpenes derived from Wedelia paludosa with the Plasmodium falciparum sarco/endoplasmic reticulum Ca²⁺-ATPase PfATP6.
作者:
主题词
抗疟药(Antimalarials);青蒿素类(Artemisinins);钙(Calcium);钙转运ATP酶类(Calcium-Transporting ATPases);二萜类, 贝壳杉烷(Diterpenes, Kaurane);药物设计(Drug Design);药物相互作用(Drug Interactions);酶抑制剂(Enzyme Inhibitors);分子结构(Molecular Structure);恶性疟原虫(Plasmodium falciparum);肌浆网钙转运ATP酶类(Sarcoplasmic Reticulum Calcium-Transporting ATPases);毒胡萝卜内酯(Thapsigargin);蟛蜞菊属(Wedelia)
DOI
10.1590/0074-02760140415
PMID
25946251
发布时间
2021-09-15
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