Synthesis and in vitro evaluation of [18F]FECIMBI-36: A potential agonist PET ligand for 5-HT2A/2C receptors.
第一作者:
Jaya,Prabhakaran
第一单位:
Department of Psychiatry, Columbia University College of Physicians and Surgeons, New York, NY, USA. Electronic address: jp2155@cumc.columbia.edu.
作者:
医学主题词
剂量效应关系, 药物(Dose-Response Relationship, Drug);乙胺类(Ethylamines);氟放射性同位素(Fluorine Radioisotopes);人类(Humans);配体(Ligands);分子结构(Molecular Structure);正电子发射断层显像术(Positron-Emission Tomography);受体, 血清素, 5-HT2A(Receptor, Serotonin, 5-HT2A);受体, 血清素, 5-HT2C(Receptor, Serotonin, 5-HT2C);血清素5-HT2受体激动剂(Serotonin 5-HT2 Receptor Agonists);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bmcl.2015.07.034
PMID
26253634
发布时间
2020-11-17
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