Recognizing drug targets using evolutionary information: implications for repurposing FDA-approved drugs against Mycobacterium tuberculosis H37Rv.
第一作者:
Gayatri,Ramakrishnan
第一单位:
Indian Institute of Science Mathematics Initiative, Indian Institute of Science, Bangalore-560012, India and Molecular Biophysics Unit, Indian Institute of Science, Bangalore-560012, India. ns@mbu.iisc.ernet.in.
作者:
医学主题词
氨基酸序列(Amino Acid Sequence);抗结核药(Antitubercular Agents);细菌蛋白质类(Bacterial Proteins);结合部位(Binding Sites);计算生物学(Computational Biology);药物设计(Drug Design);药物重新定位(Drug Repositioning);人类(Humans);模型, 分子(Models, Molecular);分子构象(Molecular Conformation);分子序列数据(Molecular Sequence Data);结核分枝杆菌(Mycobacterium tuberculosis);蛋白质结合(Protein Binding);序列比对(Sequence Alignment);构效关系(Structure-Activity Relationship)
DOI
10.1039/c5mb00476d
PMID
26429199
发布时间
2015-11-11
- 浏览14
Molecular bioSystems
3316-31页
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