Advantages and Challenges of Phenotypic Screens: The Identification of Two Novel Antifungal Geranylgeranyltransferase I Inhibitors.
作者:
主题词
烷基和芳基转移酶类(Alkyl and Aryl Transferases);抗真菌药(Antifungal Agents);药物发现(Drug Discovery);抗药性, 真菌(Drug Resistance, Fungal);酶抑制剂(Enzyme Inhibitors);基因表达谱(Gene Expression Profiling);代谢组学(Metabolomics);微生物敏感性试验(Microbial Sensitivity Tests);模型, 分子(Models, Molecular);分子构象(Molecular Conformation);突变(Mutation);蛋白质结合(Protein Binding);酿酒酵母菌(Saccharomyces cerevisiae)
DOI
10.1177/1087057115610488
PMID
26459507
发布时间
2016-12-30
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