6-Methylpurine derived sugar modified nucleosides: Synthesis and in vivo antitumor activity in D54 tumor expressing M64V-Escherichia coli purine nucleoside phosphorylase.
第一作者:
Abdalla E A,Hassan
第一单位:
Southern Research Institute, P.O. Box 55305, Birmingham, AL, 35255-5305, USA; Applied Nucleic Acids Research Centre, Zagazig University, Zagazig, PO Box 44519, Egypt. Electronic address: abdallaelsayed@zu.edu.eg.
作者:
主题词
动物(Animals);抗肿瘤药(Antineoplastic Agents);碳水化合物(Carbohydrates);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);酶抑制剂(Enzyme Inhibitors);大肠杆菌(Escherichia coli);人类(Humans);小鼠(Mice);分子结构(Molecular Structure);肿瘤, 实验性(Neoplasms, Experimental);核苷类(Nucleosides);嘌呤核苷磷酸化酶(Purine-Nucleoside Phosphorylase);嘌呤类(Purines);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.ejmech.2015.12.029
PMID
26724729
发布时间
2017-07-26
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