Synthesis, Biological, and Computational Evaluation of Substituted 1-(2-Methoxyphenyl)-4-(1-phenethylpiperidin-4-yl)piperazines and 1-(2-Methoxyphenyl)-4-[(1-phenethylpiperidin-4-yl)methyl]piperazines as Dopaminergic Ligands.
作者:
主题词
动物(Animals);结合部位(Binding Sites);多巴胺(Dopamine);多巴胺药(Dopamine Agents);药物设计(Drug Design);配体(Ligands);男(雄)性(Male);分子动力学模拟(Molecular Dynamics Simulation);哌嗪类(Piperazines);蛋白质结合(Protein Binding);大鼠(Rats);大鼠, Wistar(Rats, Wistar);受体, 多巴胺D2(Receptors, Dopamine D2);构效关系(Structure-Activity Relationship)
DOI
10.1002/ardp.201600081
PMID
27335270
发布时间
2017-03-02
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Archiv der Pharmazie
614-26页
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